Fioricet® (Butalbital, Acetaminophen, and Caffeine Tablets USP) is supplied in tablet form for oral administration.
Each tablet contains the following active ingredients:
butalbital USP . . . . . . . . . . . .50 mg
acetaminophen USP . . . . . . 325 mg
caffeine USP . . . . . . . . . . . . .40 mg
Butalbital (5-allyl-5-isobutylbarbituric acid), is a short to intermediate-acting barbiturate. It has the following structural formula:
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C11H16N2O3 Mol. wt. 224.26
Acetaminophen (4´-hydroxyacetanilide), is a non-opiate, non-salicylate analgesic and antipyretic. It has the following structural formula:
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C8H9NO2 Mol. wt. 151.17
Caffeine (1,3,7-trimethylxanthine), is a central nervous system stimulant. It has the following structural formula:
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C8H10N4O2 Mol. wt. 194.19